Neurokinin Receptor Inhibitors

NK1R

NK2R

NK3R

Neurokinin Receptor Inhibitors, Agonists, Antagonists & Modulators

Product Name	NK1R	NK2R	NK3R	Purity
Substance P	NK1R			99.60%
Senktide	NK1R, EC₅₀: 35 nM		NK3R, EC₅₀: 0.5-3 nM	99.91%
Fezolinetant			NK3R	99.19%
EB1002		NK2R		99.98%
L-659874		Hamster Bladder NK-2, IC₅₀: 0.49 μM
Ranakinin	NK1R
Rolapitant	human NK1, Ki: 0.66 nM gerbil NK1, Ki: 0.13 nM guinea pig NK1, Ki: 0.72 nM monkey NK1, Ki: 2.5 nM rabbit NK1, Ki: 31.7 nM rat NK1, Ki: 78.6 nM mouse NK1, Ki: 60.4 nM			99.89%
N-Acetyl-L-tryptophan	NK1R			99.82%
Saredutant		NK2R		98.09%
SB-222200			NK3R	99.85%
L-733060 hydrochloride	NK1R			99.9%
GR-73632	NK1R			99.89%
L-732138	NK1R, IC₅₀: 2.3 nM			99.9%
Substance P TFA	NK1R			99.34%
Pavinetant			NK3R	99.63%
Talnetant			NK3R	99.38%
Osanetant			NK3R	98.19%
Orvepitant maleate	NK1R, pKi: 10.2			99.99%
Eprazinone dihydrochloride	NK1R			99.05%
GR 159897		hNK2, pKi: 9.51 (CHO cell) NK2R, pKi: 10 (Rat colon membrane)		99.60%
Vapreotide	NK1R			99.72%
Spantide II	NK1R			99.47%
Biotin-Substance P	NK1R			99.66%
Casopitant mesylate	NK1R			99.83%
Spantide I	NK1R, Ki: 230 nM	NK2R, Ki: 8150 nM		99.64%
Maropitant	NK1R			99.39%
[Lys5,MeLeu9,Nle10]Neurokinin A(4-10)		NK2R		99.89%
Vofopitant dihydrochloride	NK1R, pKi: 9.02			99.56%
GR 64349		NK2R		99.12%
Eledoisin		NK2R	NK3R	99.06%
Rolapitant hydrochloride hydrate	human NK1, Ki: 0.66 nM gerbil NK1, Ki: 0.13 nM guinea pig NK1, Ki: 0.72 nM monkey NK1, Ki: 2.5 nM rabbit NK1, Ki: 31.7 nM rat NK1, Ki: 78.6 nM mouse NK1, Ki: 60.4 nM			98.36%
Hemokinin 1 (mouse)	NK1R			98.38%
Vapreotide acetate	NK1R			99.85%
NKP608	NK1R, IC₅₀: 2.6 nM			99.88%
MEN 10207	NK1R, pA2: 5.2	Tachykinin NK₂ Receptor, pA2: 7.9	NK3R, pA2: 4.9	99.80%
[MePhe7]-Neurokinin B			NK3R, IC₅₀: 3 nM	98.76%
Fosnetupitant chloride monohydrochloride	hNK1, pKi: 9.5		hNK3, pKi: 6.1	99.70%
Vofopitant	NK1R, pKi: 9.02			99.82%
Hemokinin 1, human	NK1R	NK2R	NK3R	98.11%
Nolpitantium	NK1R
γ-Neuropeptide (rabbit)		NK2R		99.99%
L-760735	hNK1, IC₅₀: 0.19 nM			99.9%
SB 218795		hNK2, Ki: 1220 nM	hNK3, Ki: 13 nM	99.86%
SCH-720881	NK1R
SDZ NKT 343	hNK1, IC₅₀: 0.62 nM	hNK2, Ki: 0.52 μM	hNK3, Ki: 3.4 μM
Hemokinin 1, human TFA	NK1R	NK2R	NK3R
CS-003 Free base	NK1R, Ki: 2.3 nM	NK2R, Ki: 0.54 nM	NK3R, Ki: 0.74 nM
(Trp7,β-Ala8)-Neurokinin A (4-10)			NK3R
Scyliorhinin I	rat NK1, Ki: 0.9 nM	guinea pig NK-2, Ki: 2 nM
MDL 105212A	NK1R	NK2R
[D-Trp2,7,9] Substance P	NK1R, Ki: 1 μM	NK2R, Ki: 1.3 μM	NK3R, Ki: ~9 μM
[S5K, F6Y, L9mL, M10Mox] neurokinin A (4-10)	NK1R			98.14%
GR 94800 TFA		NK2R
CP-99994 hydrochloride	NK1R, Ki: 0.25 nM
GR 64349 acetate		NK2R
NK3R-IN-2			NK3R
Senktide TFA	NK1R, EC₅₀: 35 μM		NK3R, EC₅₀: 0.5-3 nM
NK3R antagonist-1			NK3R, IC₅₀: 53.61 nM
MEN 10207 acetate		NK2R
SB 414240		hNK2, Ki: 1 nM	hNK3, Ki: 193 nM
Phyllomedusin	NK1R
GR 64349 TFA		NK2R
Imnopitant	NK1R
L-741671	hNK1, Ki: 0.03 nM
RO5328673		hNK2, Ki: 1.1 nM	hNK3, Ki: 0.4 nM
UK-224671		NK2R
L-733060	NK1R
TKA-731	NK1R
SSR 146977			NK3R
Rolapitant hydrochloride	human NK1, Ki: 0.66 gerbil NK1, Ki: 0.13 guinea pig NK1, Ki: 0.72 monkey NK1, Ki: 2.5 rabbit NK1, Ki: 31.7 rat NK1, Ki: 78.6 mouse NK1, Ki: 60.4
Neurokinin Receptor (393-407), rat	NK1R
CP 122721 hydrochloride	human NK1, pIC₅₀: 9.8
[Lys5,Tyr6,mLeu9,Nle10]-Neurokinin A (4-10)		hNK2, EC₅₀: 3.7 nM	hNK3, EC₅₀: 450-3500 nM
Benzomalvin A	NK1R
Acetylaszonalenin	NK1R
GSK256471			NK3R, pIC₅₀: 8.9
(D-Arg1,D-Pro2,D-Phe7,D-His9)-Substance P	NK1R
ASN-1377642	NK1R, Ki: 251 nM
[Pro9]-Substance P	NK1R, EC₅₀: 0.93 nM
CP-99994	NK1R, Ki: 0.25 nM
DNK-333	NK1R, pkB: 9.2 hNK1, IC₅₀: 4.8 nM	NK2R, pkB: 7.43 hNK2, IC₅₀: 5.5 nM
Vestipitant mesylate	human NK1, pKi: 9.65
GR 87389		NK2R
[Asp5,6,Me-Phe8] Substance P (5-11)			NK3R
Telmapitant	NK1R
TAC 363		Tachykinin NK₂ Receptor, pA2: 9.82
GSK172981			hNK3, pKi: 7.7 Native guinea pig NK3, pKi: 7.8
WIN-64821	NK1R, Ki: 0.24 μM	NK2R, Ki: 0.26 μM	NK3R, Ki: 15.2 μM
Maropitant citrate	NK1R
YM-49598 iodide	NK1R
Vestipitant	hNK1, pKi: 9.4
ZM 253270		Hamster Bladder NK-2, Ki: 2 nM
Befetupitant	NK1R
Fosrolapitant	NK1R
Talnetant hydrochloride			NK3R
Physalaemin	NK1R
MEN11467	NK1R

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